UtanoGadziriro

The mushonga "Triftazin": mirayiridzo kushandiswa, mutengo, analogs, wongororo. Ovhadhozi, marwadzo, uye abolition kuti "triftazin"

Drug "Triftazin" mirayiridzo chichakurukurwa zvakajeka muna ino, runoonekwa mumwe inonyatsobudirira antipsychotic mishonga. Kushandiswa kwezvinodhaka iri chokuita subtleties zhinji panyaya chipimo chemushonga uye nguva yokurapa.

Description rekugadzirira, akafanana

Maererano boka chavanopinda zvinodhaka "Triftazin" rinoreva simba antipsychotic mushonga ane raidudzwa Anti-emetic mugumisiro. The chikuru kushingaira chirungiso ndiyo remubatanidzwa kubva boka phenothiazines - trifluoperazine, izvo zvinogona kukanganisa musimboti tsinga, asiwo kwayo peripheral Zvikamu, saka, chokwadi, ane antiemetic mugumisiro.

A mhinduro jekiseni riri pachena, Hauoneki mvura, hapana kunhuwa yaingowanikwa uye kuravira. Mahwendefa "Triftazin" vakagumisa, zvemapuranga yebhuruu, pakutanga kwezana chena kana anenge chena.

Release chimiro, mashoko uye mamiriro ezvinhu okuchengetera

Medicine "Triftazin" apindure vanachiremba pamusoro dzinenge nguva dzose akanaka, rinowanika zviviri chipimo chemushonga siyana: sezvo kugadzirisa kuti jekiseni uye mahwendefa. Zviri vanoshingaira fuma neimwe ampule ine mhinduro ine 0.2% (2 MG muna 1 Rine mamiririta mhinduro). The ampoules vari mumapepa makatoni pa 5, 10, kana 100 zvidimbu pamwe rinokosha ampoule banga uye mirayiridzo kushandiswa kwezvinodhaka.

Pamahwandefa "Triftazin" zvinoshingaira fuma zvirimowo mune mari 0,005% (0.5 MG). Ivo vari kugara mu Maronda akasiyana zvezvimedu 10, izvo, akavapindurawo, akaisa mumabhokisi makadhibhokisi pamwe 4, 5 kana 10 zvidimbu nerimwe. Uyewo iripo chipimo chemushonga chimiro mumidziyo rima negirazi kana chichena opaque mupurasitiki, ine mahwendefa 50 kana 100.

Pasherufu upenyu zvose chipimo chemushonga siyana zviri 3 years. Vanounganidza mapiritsi uye mhinduro "Triftazin" mirayiridzo kushandiswa anokurudzirwa inotonhorera nzvimbo ine kufefetedza zvakanaka. Haugoni kubvumira kuti Mabhokisi mishonga kutungamirira chiedza chezuva kana mvura mvura. haina yakarumbidza kutora mushonga mushure expiry musi.

Pharmacological ehupfumi "Triftazin" chinodhaka

Ngatikurukurei dzinokosha ehupfumi zvinodhaka "Triftazin". Mirayiridzo kushandiswa (mukuru) rinonyatsotsanangura ruzivo pamusoro mashandiro chiito yezviri zvinodhaka fuma kune receptors muuropi uye ari vagus etsinga ari gastro-intestinal turakiti. Somuenzaniso, rinotaura kuti trifluoperazine PMD kutigumbura receptors muuropi uye D2 receptors ari cerebellum. Kunze neuroleptic ichi vanokwanisa kupa munhu Arufa-adrenoceptor ichivharira kushanda, kureva, kushingaira simba pamusoro BP, richikwidibira nayo.

Zvisinei Trifluoperazin akadzidza zvikuru zvakakwana maererano pharmacokinetics,, achinyatsoziva kuti akanga ari kushingaira vakasungwa mapuroteni eplasma (kanenge 80%). kuora coupling nomazviri metabolites sezvo ambodzidza nezvishoma. Excretion zvinodhaka kubva muviri kunoitika kunonyanya nomukombiyuta itsvo, chikamu chiduku yezviri fuma uye metabolites waro goho kuburikidza ura (mu bile).

zvairatidza

Sezvo chiito "Triftazin" gadziriro kudzidziswa Chinyorwa classifies sezvo antipsychotic, zvakawanda zvirwere nokuti icho Zvakakunakirai kushandisa, rinosanganisira dzakasiyana-siyana chirwere chepfungwa. Pakati pavo - schizophrenia, psychomotor nenyonganiso, kufunganya uye phobias (chin'a nyanyisa kutya). Kunze mushonga unoshandiswa kuti kurapa emesis hazvikonzerwi gastrointestinal zvirwere.

wakachengeteka sei tiri kufunga nzira uye kana Mapato ose varwere vanogona kushandiswa "Triftazin"? Mirayiridzo yokushandisa, nyanzvi chaiwo zvinganzi kwakagumisa kuti zvakakosha kutora mushonga chete pashure ichiitwa misoro kuongorora, sezvo ane vanoverengeka chakakomba nemishonga uye contraindications. Pasinei chokwadi kuti zvakabudisa mushonga pasina mushonga, kuti kusarudza kubvuma kwake hakusi zvakakodzera.

Contraindications

At mahwendefa uye mhinduro kuti "Triftazin" majekiseni ndivo contraindications kushandisa kuti inotaura hazviiti avo kushandiswa. Pakati pavo vanonzi nechepakati tsinga mwoyo uye pakoma. Mukuwedzera, zvinodhaka "mirayiridzo Triftazin 'kushandiswa haina akakurudzira kutora nezvirwere zvomwoyo, chiropa uye itsvo, hematopoietic hurongwa. Pavaipfuura chirwere uye kukuvadza kwayo kosi asingadi kuita basa rinokosha. Yokuti pane wandei migumisiro negashiro mahwendefa uye "Triftazin" mhinduro. Marwadzo, iyo ichakurukurwa Papera, pachavo vari rinorema kwazvo, uye kuvapo comorbidities anogona kutsamwisa zvakatonyanya kuoma migumisiro murwere.

Zvinonzi Dzakamukurudzirawo haana kushandisa mudziyo ane nhoroondo neutachiona upi chikamu zvinodhaka.

Uchishandisa "Triftazin" panguva pamuviri

The vanoshingaira fuma mishonga "Triftazin" (wongororo vanachiremba ane nezvazvo yakawanda yokutsigira mashoko) inokanganisa pamusoro kukura azvarwa. Zvinonzi saka haana yakarumbidza kutora mushonga panguva yepamuviri. Chokwadi chokuti basa fuma trifluoperazine dzakaonekwa mune fetus nyama iri kuwanda yakakwirira zvikuru kupfuura kuchirapa mishonga. Kuti chinokurwadzai simba akagadzirwa fetus uremu, uye kuwedzera ngozi urema siyana ari kukura kwake.

Drug "Triftazin" (analogs yezviri fuma Zvinokoshawo kufunga) haina varumbidzwa uye lactating vakadzi zvinodhaka zvinhu zvinowanikwa mukaka. Kunyange kana amai kana kurinda chero divi migumisiro, mwana ramangwana vangasangana nematambudziko akadai tardive dyskinesia uye nokuvhiringidzika.

nemishonga

Sezvambotaurwa, mushonga "Triftazin" kunogona kukonzera zvinoverengeka nenjodzi pamusoro chikamu zvinenge zvose nhengo uye hurongwa. Zvikurukuru kushingaira fuma kunokanganisa tsinga murwere, izvo zvinoreva kuti mugove divi anokonzerwa weshumba rinowanika mairi. Chokutanga, zvinosanganisira zviitiko zvakadai chakamira pakunodengenyeka zvine, kwetsandanyama kwemitsipa uye mutauro, nei anogona kunokanganisika (extrapyramidal siyana). zviratidzo tardive dyskinesia kuonekwa sezvo kazhinji, kushaya hope, akathisia, uye autonomic zvirwere.

Rakajairika nenjodzi kubva nechepakati tsinga anokonzerwa yaunodya kuti "Triftazin" chinodhaka mhinduro anonzi hope, dzungu uye kurasikirwa zvakajeka wezvakaonekwa. Kazhinji Zviratidzo izvi zvichiitika mukati rokutanga pashure pakatanga kurapika.

Chiizve kunogona kukonzera panosvikira mhinduro kuti jekiseni kana mahwendefa "Triftazin"? Nemishonga, maererano neuchapupu kuvarwere uye vanachiremba, kazhinji zvinokanganisa zvomudumbu hurongwa. Izvi zvinoonekwa muchimiro mumuromo yakaoma uye neanorexia. Uyewo, kazhinji pane nezvinetso chakaipa nokushanda kwenhengo chiropa. Mukuwedzera, pangava nechitarisiko sema ganda mapundu, amenorrhea, agranulocytosis.

Zvokungwarira

Zvataurwa pamusoro apa nemigumisiro zvinogona mitigated nokuda symptomatic kurapwa kana dose kuchinja. Kukanzura "triftazin" kunodiwa chete kana paine chakakomba Kuvhiringidza kuti murwere nenhengo dzawo. Saka, isu funga dzinokosha unyanzvi uye nzira kwetsvina kana kuderedza kuti pasingadiwi anwa mushonga.

Kana chakamira pakunodengenyeka zvine kana pfari kazhinji, nyanzvi vari kusarudza kuderedza mishonga rakatorwa murwere kana kwekanguva kumira mutambo wake. In kwazvo Muzviitiko kungada kurapwa pamwe antiparkinsonian zvinodhaka, barbiturates kana zvine caffeine zvinodhaka (intravenous yaitonga).

Apo akazivisa zviratidzo hope kana injini disinhibition, kushungurudzika haisi yakarumbidza kuwedzera pokutangira dose. Kazhinji mumazuva mashomanana muviri zvinoenderana kuti mushonga mutsva, uye yaivhuvhuta zviratidzo zvishoma nezvishoma kunyangarika. Zvikasadaro, kungada kurapwa zvinodhaka "benzodiazepine" kana "Propanolol".

mamiriro akadaro tardive dyskinesia, ambotaurwa pakati nemishonga kana achitora "Triftazin" chinodhaka, wongororo izvo zvichaita kunzi hereinafter, kazhinji achikura zvichikonzerwa kushandiswa kwezvinodhaka kana nguva pfupi pashure ayo kukanzura-refu. Nyanzvi dzinoti dyskinesia (tardive) anowanzodanwa chirwere Varwere vakwegura.

Vamwe divi matambudziko anokonzerwa yaunodya ane medicament kuchipesana nokusava zviito akadai kudzora motokari uye zvakaoma zvigadziriswe. Panguva kurapwa "triftazin" nani kurega kwavari.

Matungamirire dosages uye nzira gadziriro Hour

Chipimo chemushonga pakutsvaga nyanzvi pahwaro wacho murwere, ake ezvinhu uye kuvapo concomitant zvirwere. Minimum dose "Triftazin" mushonga kakawanda chinotarisirwa mukutanga nzira yokurapa. Mahwendefa kurairira anorayiridza kutora 1-5 MG 2 kanomwe pazuva (varwere mukuru). Mumakore akatevera nhatu, kuti chipimo chemushonga ichiwedzerwa zvishoma nezvishoma uye kumamiriro 45-60 MG pazuva. mari iyi anofanira kukamurwa muzvikamu zvitatu.

Nokuti kurapa vana zvakajairika kushandisa mishonga diki zvinodhaka. Pakutanga kurapwa musatora kupfuura 3 MG pazuva (muna 3 mumatanho). Kana zvakakodzera, uye pasina raidudzwa divi anokonzerwa Zviratidzo zviri dose yakanga yawedzera kusvika 6,5 MG pazuva.

Jekiseni "Triftazin" anofanira kuzviita intramuscularly pane zvikamu kwete kupfuura 6 maawa. The dose zuva nezuva vakuru vane vaifanira 10 MG. Babies inoratidza chipimo chemushonga 1 MG pazuva, rakakamurwa majekiseni maviri, pane zvikamu kwete asingasviki 12 maawa.

Tinoswedera muverengi afunge kuti kurapwa pamwe zvinodhaka ichi, pasinei chipimo chemushonga fomu yaifanira pasi pokudzora chiremba. Ndiye anosarudza pamusoro chipimo chemushonga kuchinja mishonga kusarudza "Triftazin". Ovhadhozi kana ikashandiswa zvakanaka, zvinoreva kutonetsa. Kunze komutemo kushandiswa kwezvinodhaka, kana kuchinja zvavakabvumirana dose hombe nzira kungaita kuti nezvimwewo nemigumisiro.

zvinodhaka kwavatori

mishonga All vanowanzoda kushamwaridzana nomumwe. Mahwendefa uye "Triftazin" jekiseni munaizvozvo kuvapowo. Kazhinji, vanachiremba kufungawo zvinhu zvakawanda kuti kukanganisa kunyatsoshanda kuti kushandisa zvinodhaka ichi. Saka, medicaments rine panyaya iyi (syrups, neiya inoiswa muzvinwiwa zvinodhaka uye zvakafanana), CNS kuora mwoyo kunogona kuwedzera zvivako zviri "triftazin", uyewo kukanganisa mashoko dzinotsanagura afemeruke.

Pachiimbwa zvinodhaka izvo kuderedza BP, pokunyorera kana mhinduro "Triftazin" rinofanira kuiswa vanyatsohuongorora sezvinobvira kukura chakasimba orthostatic hypotension.

Antacids uye antiparkinsonian yomuchipatara zvinobatsira muduku Absorção de Água yezviri fuma pellets "Triftazin" kubva zvomudumbu turakiti uye, saka, kuderedza kubudirira chezvinodhaka.

The kunambwa kunoonekwa uye kana mushandirapamwe vakashandisa zvinodhaka lithium munyu. Maererano mashoko akapiwa, zvakadai mubatanidzwa hwakazara Kugadzirwa raidudzwa extrapyramidal zviratidzo uye kwakawedzera neurotoxic mugumisiro trifluoperazine.

Reviews zvokurapa "Triftazin"

vazhinji vari kuedza kuwana wongororo nezvazvo usati watanga achitora zvinodhaka. Medicine "Triftazin", kutonga nezvinooneka zvakataurwa nenyanzvi, runoonekwa mumwe inonyatsobudirira. Panguva iyoyowo, ivo cherechedza kuti inondimukira achitora mushonga angava inokanganisa kwete chete pane mumuviri asi epfungwa wemunhu.

Nokuti avo varwere vakaratidza negashiro zvinodhaka, kakawanda kacho ndiyo chete nzira kurarama sezvinongoita. Chokwadi, hakusi pasina nemishonga. Asi, maererano nenhamba, zvose zvinoitika zviratidzo inonyangarika mukati vaifanira vhiki mbiri pashure mharuro mushonga.

Maonero pamusoro dzevarwere Triftazin "mushonga yakavhenganiswa. Mumwe akabatsira chaizvo, nepo vamwe vari saka zvakaoma kushivirira marwadzo kuti vaifanira kusiya chokushandisa ichi. Kakawanda vatengi anoratidza nechitarisiko kuneta, lethargy uye mukuru muutera. Mune zvisingawanzoitiki Muzviitiko, varwere nehope mamiriro apo havadi kuita kunyange inokosha kufamba.

Women, kusiyana nevanhu, vari kazhinji kutaurwa kuwedzera uremu muviri panguva kurapwa ne "Triftazin". Nyanzvi vanoti kwainge pakati kurapa ichi zvinodhaka uye hapana kufuta. Vaifunga kuti izvi imhaka vasanyanye injini basa varwere tikafunga nokuchengetedzwa aimbova kudya.

Dzakakurudzira panyaya mugumisiro zvinodhaka, uye vanachiremba uye varwere vakaona kuti chaizvoizvo hwezvekukurukurirana kana anobvisa zvose zviratidzo runotikurudzira chirwere.

Analogs uye Mari zvinodhaka

Saka, isu akaongorora pezvidzidzo pakushandisa "Triftazin" chinodhaka. Imomo mune nayo rinoenderana kutsiva, kana inonzi analogs? Chokwadi, zvinodhaka izvi zviuru. Antipsychotics zvava kubudisa chinenge zvose nemakambani anogadzira mishonga, uye vakawanda zvinodhaka muboka iri dzinoturwa zvakafanana "triftazin" (kureva kusangana naye pamusoro murwiyo). Izvi zvinosanganisira "Vespezin" zvinodhaka "trifluoperazine hydrochloride", "trifluoperazine hydrochloride", "fluazinam," "Ekvazin", "Stelazin", "Cyclodol" uye vamwe vakawanda.

Mari zvinodhaka izvi hazvisi zvakafanana nguva dzose. Foreign dzomuzana kakawanda zvinodhura, zvichienzaniswa zvinodhaka "Triftazin", mutengo avhareji 50-70 rubles por rongedza (Mahwendefa 50). Kana tikafunga kuti nokushandiswa chokushandisa ichi, nguva yokurapa, anogona kunzi kukosha kwayo somumwe huru zvakanakira pamusoro dzimwe analogs.

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