UtanoGadziriro

The mushonga "papaverine" (kwepfuti)

Medicament "papaverine" (majekiseni) ndiro antispasmodic, vane hypotensive migumisiro. The mushonga anokwanisa tunodzivisa PDE (PDE), chikonzero kuunganidza Camp (cyclic Adenozinmonosfata) richikwidibira Ca2 +.

Rinoreva "Papaverine" (jekiseni) relaxes uye anoderedza anotsvedzerera tsandanyama mataurire zvomukati (genitourinary, zvomudumbu, kufema) nemidziyo. Inosimudzira chipimo chemushonga anogona kuderedza excitability mwoyo tsandanyama uye kunonoka conduction (intracardiac). Drug "papaverine" (kwepfuti) ane zvakaneta iziviswe zvainoita CNS. In guru mishonga ine kunyaradza simba.

Kubudirira zvinodhaka kwakacherechedzwa pashure maviri kusvika makumi mana maminitsi pashure kutarisira. Zvakaitwa zvinodhaka hunogara kubva mana nhanhatu maawa.

Rinoreva "papaverine" (majekiseni) kunoratidzwa nokuda spasm pakati anotsvedzerera tsandanyama ose peripheral vascular (endarteriite), nhengo iri abdominal mhango (renal colic, spastic colitis pilorospazme, cholecystitis), mwoyo (angina pakurapwa), midziyo uropi (chepfungwa). The mushonga zvinoratidzwa nekuda premedication (kugadzirira kuvhiyiwa) ari chikamu zvinodhaka.

Haungopiwi yemaziso, hypersensitivity, AV nechigumbuso, vakwegura, mune renal kukundikana zvikuru, pauduku (kusvika mwedzi mitanhatu).

With kunyatsogadzirira rinoshandiswa varwere vakambova musoro kunotevera, kuvhunduka ezvinhu, pamwe kukwana basa iri adrenal shwanu, hyperplasia isiri yekenza kweprostate gland, hypothyroidism, supraventricular tachycardia.

Kushandisa zvinodhaka izvi zvinogona kunyengedza ventricular arrhythmia, kupatira, BP, sema maitiro, nehope, eosinophilia, vakawedzera transaminase basa "chiropa".

In ovhadhozi akacherechedza diplopia, somnolence, utera, kuderera kumanikidza (ropa). Symptomatic kurapwa inofanira kutsigira BP.

"Papaverine" majekiseni. Mirayiridzo kushandiswa.

Subcutaneously, intramuscularly dzakabatwa maviri kusvika makumi mana milligrams (1-2 Rine mamiririta maviri muzana mhinduro), rimwe zuva, vaviri mana nguva. Intravenous jekiseni rinoitwa zvishoma nezvishoma. Chipimo chemushonga - maviri milligrams.

Kushandisa zvinodhaka "papaverine" (majekiseni) anofanira kuzviita chete pasi zvokurapa achitarisirwa.

Panguva kurapa zvakafanira kuti asava kubvuma panyaya iyi.

Akaora chigaro kuchengeteka zvinodhaka panguva yepamuviri uye lactation. Kugadzwa hauna varumbidzwa pasi izvi ezvinhu.

Kana fodya kunoderedza vasodilating medicament.

Drug "papaverine" anogona kuderedza hypotensive mugumisiro methyldopa uye levodopa antiparkinsonian efficacy. Pane amplification antispasmodic ehupfumi zvinodhaka vachishandisa pamwe barbiturates. Hypotensive mugumisiro zvinoreva anogona ngazviwedzerwe kana pamwe quinidine, reserpine, procainamide, tricyclic antidepressants.

The mushonga rinowanikwa mururimi piritsi chimiro, muchimiro suppositories. Makenduru vane munharaunda zvazvinoita. Kazhinji ivo (suppository) zvaishandiswa Gynecology kuvasunungura spastic inoti. Makenduru vanoonekwa kunoreva zvakawanda simba kuvasunungura kurwadza kwacho ari pelvic zvomukati.

Kushandisa zvinodhaka muvana vanofanira raitarisirwa nyanzvi.

Kugadzwa inofanira kudzivirira kubata pamberi contraindications.

Kubvuma nehwendefa chimiro mushonga muvana vanofanira kuongororwa pedyo mazvikokota.

Rinoreva "papaverine" anonzi zvikuru zvakajairika zvinodhaka kusimbisa kurwadza kwacho. Sezvinoratidzwa kurapwa tsika, mishonga zvakanaka akashivirira nevarwere.

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