UtanoGadziriro

"Ortanol": chii zvinobatsira, mirayiridzo kushandiswa, zvechokwadi

Chii chinodhaka "Ortanol"? Kubva chii chinobatsira mushonga? Mhinduro dzemibvunzo iyi dzinogona kuwanika pazasi. Mukuwedzera, ratinoparidza mutengo akati chigadzirwa, ayo contraindications, analogs uye kusunungura chimiro.

Kavha chinodhaka, ayo akafanana, tsananguro, chimiro

Kugadzirira "Ortanol" chakaitwa nenzira dzakaoma capsules saizi № № 1 kana 2. Izvi zvinoreva ane ruvara chena, uyewo akanyorwa «Ome 20» kana «Ome 40 '(zvichienderana chipimo chemushonga). Content somushonga capsules rinomiririra yeyero pellets.

Izvi zvinosanganisira mishonga "Ortanol"? Reviews zvinoratidza kuti zvinokosha fuma ichaongororwa zvinodhaka omeprazole. Uyewo ane ebetsero zvinoriumba zvakadai croscarmellose yavaibvisa, pasi kuchiiswa giproloza, lactose anhydrous, microcrystalline cellulose, hypromellose phthalate, povidone, polysorbate 80, talc uye dibutyl sebacate.

The Kuronga Kamudzira goko zvinosanganisira: propylene glycol, hypromellose, butanol, carrageenan, anhydrous panyaya iyi, shellac, potassium chloride, anhydrous isopropanol, titanium dioxide, ingi nokuti inscribing uye mvura.

In Kutengeswa medicament "Ortanol" (Kamudzira) anopinda mhoni, mumapepa kupinda mabhokisi makadhibhokisi.

Pharmacological zviito zvinodhaka

Chii chinonzi "Ortanol" (kubva chii anobatsira mushonga uyu, uchadzidza pazasi)? Maererano mirayiridzo, mushonga chinhu inhibitor kuti hwepurotoni pombi. It kunoderedza iine acid kugadzira, kureva, DZEMUNHU DZINODZORA basa K + -H + -ATPase mudumbu, kana pane ari parietal mumasero ake. Uyewo Zvidhinha kwokupedzisira padariro gastric asidhi secretion.

Drug "Ortanol", mitengo iri pasi apa, ane prodrug. chokushandisa Izvi kusashanda ari acidic svikiro iri tubules (secretory) parietal masero. Uyezve, kunoderedza dzinovhurika uye basal secretion zvisinei yezvakaita vakurukurirane.

Antisecretory ehupfumi of medicament kuitika mukati maminitsi 60 okutanga (kunonyanyisa pashure 2 maawa). Chinovhiringidza 50% of kunonyanyisa secretion mberi yose zuva.

A chete dose of zvinodhaka zvinopa runziro uye kukurumidza kudzvinyirira kuti usiku uye masikati gastric secretion. kunonyanyisa kwayo anosvika 4th zuva kurapwa uye inonyangarika pashure pemazuva matatu pashure kurapwa.

Kinetic ehupfumi zvinodhaka

Pamusoro pokugamuchira "Ortanol" gadziriro nayo inowana kumusoro Absorção de Água. Peak kuwanda omeprazole muropa vakachengeta pashure pemaawa 0.5-3. The Mhedziso bioavailability zvinodhaka riri 30-40%, uye medicament chokuita mapuroteni eplasma - 95%.

Omeprazole muviri ari chiropa yokuumba nhanhatu pharmacologically basa nomukaka.

The hafu-upenyu mishonga nguva yava maawa 0.5-1. Output nayo sezvo nomukaka kubudikidza itsvo (70-76%) uye pamwe chete bile (18-24%).

Vanhu vane chirwere chiropa nezvirwere bioavailability zvinodhaka zviri kwakawedzera, uye plasma hafu-upenyu rinosvika maawa 3.

In varwere chirwere cheitsvo excretion DZEMUNHU DZINODZORA. Izvi kunoitika maererano zvinoderedza CC.

Medicament "Ortanol": chii zvinobatsira?

Viewed kugadzirira zvinoratidzwa zvokushandisa zvinotevera zvirwere:

  • reflux esophagitis;
  • gastrointestinal urikanwi chirwere miviri (kusanganisira Kudzivirira kuitazve);
  • hypersecretory inoti (kunetseka nemaronda ari ura, Zollinger-Ellison urwere, systemic mastocytosis, polyendocrine adenomatosis);
  • yokupedza nayo Helicobacter pylori neutachiona varwere maronda chirwere ari zvomudumbu turakiti (yakasanganiswa kurapa);

  • kurapwa uye kudzivirira gastrointestinal mucosal kukuvadzwa nhengo izvo zvakakonzera NSAID (mucosal kukurwa kwevhu, dyspepsia, peptic urikanwi).

Kurambidzwa kushandiswa zvinodhaka

Ndezvipi contraindications zvinodhaka ane "Ortanol" (kubva chii chinoita chokushandisa ichi, hatina kuudzwa apa)? Maererano mirayiridzo, vaiona mushonga hazvigoni kushandiswa kana:

  • lactation;
  • yomwana;
  • hypersensitivity kuti zvinodhaka fuma.

Nokungwarira vaiona chinokosha zvinodhaka nachiremba renal uye chiropa kukundikana.

Drug "Ortanol": okuti

mushonga uyu ushandiswe chete mukati. Rakundwa asati zvokudya (kazhinji mangwanani pamberi kwemangwanani).

The Kamudzira ane mushonga vakamedzwa chose nemvura. Pakadaro, kana murwere haakwanisi kushandisa mishonga zvachose, zvirimo unogona zvazvichanyungudutswa chiduku haisi acidic chaizvo mvura.

The chipimo chemushonga zvinodhaka kunobva uchapupu.

Kana nemaronda 12 duodenal urikanwi medicament chinotarisirwa pa 20 MG kamwe pazuva kwevhiki mbiri. Kuri kuti pashure rokutanga gore rakakwana scarring hakuitiki, kuzodzosera vakagadzwa-vhiki mbiri kurapa.

In maronda chirwere husingakwanisi kurapwa, mumiririri uyu inokurudzirwa kutora chipimo chemushonga 40 MG kamwe pazuva. Nzira yokurapa pamwe zvinodhaka izvi anogona kuratidzirwa masvondo mana.

Capsules "Ortanol" zvairatidza zvakatendeka pamusoro apa, maronda maronda mudumbu achitora 20 MG kamwe zuva nezuva kwemavhiki mana. Kana scarring hariwanikwi mushure vakayambuka gore, kuti apiwa vakagadzwa-vhiki mana kurapa. In gastric urikanwi, husingakwanisi kurapwa, mishonga inokurudzirwa kutora dose 40 MG kamwe pazuva (mwero anosvika masere mumasvondo).

Yokupedza nayo Helicobacter pylori riri kuitwa mubatanidzwa mishonga. Panyaya iyi, iyo medicament chinotarisirwa pa 20 MG kaviri pazuva pamberi zvokudya (kwevhiki mbiri) akabatana antibacterial nevamiririri.

Kana reflux esophagitis zvinodhaka inokurudzirwa kushandisa mari 20 MG (kamwe) kwevhiki ina. Kana nzira iri mushonga haakonzeri kupedza mushonga, murwere ushandiswe yechipiri kosi (masvondo mana). In zvakakomba reflux esophagitis kurapwa chokushandisa ichi chinoshanda kusvika masere mavhiki.

Kana hypersecretory mamiriro kunoonekwa sechinhu mushonga chirungurira raitongwa nomumwe. Zvavakabvumirana kutanga chipimo chemushonga kuti vakuru 60 MG (kamwe), uye kufadza - 120 MG.

In agadza mushonga anopfuura 80 MG pazuva, rakakamurwa muzvikamu akawanda.

Kana kukuvara gastrointestinal mucosa nhengo, izvo zvinokonzerwa NSAID, uyewo kudzivirira Kamudzira "Ortanol" kutokurudzira kushandisa dose 20 MG ose zuva, vasati kwamangwanani (nokuti yose ya NSAID mishonga).

Nokuti vanhu vakwegura uye vanhu zvikuru chiropa chirwere kunonyanyisa daily dose ndiyo 20 MG.

Nokuti varwere havachanyatsogoni itsvo basa chipimo chemushonga kuchinja kunodiwa.

zvakavapo divi

Chii Maitiro kunaka kukonzera zvinodhaka "Ortanol"? Reviews vachiti marwadzo:

  • nemusoro, madzerere, anzwe dzungu, erythema multiforme, paresthesia;
  • Hope, kuda kurutsa, kuravira chinovanetsa, manyoka, kushaya hope, flatulence;
  • nokusagadzikana, muromo yakaoma, kuora mwoyo, chirwere, reversible mupfungwa kuvhiringidzika;
  • encephalopathy, gynecomastia, hepatitis, peripheral edema, kurutsa, uye photosensitivity;
  • abdominal marwadzo, thrombocytopenia, kupatira, pancytopenia, nokuwedzera alkaline phosphatase basa uye chiropa transaminase;
  • itchy ganda, havachanyatsogoni chiropa basa, tsandanyama simba, paumbwe gastric glandular cysts;
  • alopecia, eosinophilia, wakawedzera vangadikitira, bronchospasm, agranulocytosis, angioedema;
  • leukopenia, myalgia, fivha, arthralgia, anaphylactoid siyana, urticaria, interstitial nephritis.

Nemishonga kuti kuitika pokushandisa nhau nevasori vari munyoro uye zvinopfuura zvakasikwa.

zviitiko ovhadhozi

Kana kutora mushonga chirungurira mune murwere anotevera zvingaratidza kuitika: nemusoro, muromo yakaoma, tachycardia, hope, kuda kurutsa, madzerere, kurutsa, kuvhiringidzika, zvakawedzera iratidzike seiri kubuda.

Mumamiriro ezvinhu akadaro, symptomatic kurapa.

zvinodhaka kwavatori

Pamwechete kubvuma omeprazole yakawedzera hafu-upenyu uye kwakawedzera yevasungwa "Diazepam", "warfarin", "phenytoin", uyewo zvimwe zvinodhaka kuti rinoita iri chiropa pamwe isoenzyme CYP2C19.

Absorção de Água zvinoreva anogona anetseka, iro bioavailability uko pakutsvaga acidity pamusoro gastric muto (semuenzaniso, "Itraconazole" "ketoconazole" esters kuti ampicillin "cyanocobalamin" uye munyu simbi).

The bioavailability pamusoro digoxin kana co-raitongwa pamwe omeprazole iri yakawedzera 10%.

Viewed chinodhaka runogonesa kuti inhibitory zvainoita maitiro mamwe hematopoietic zvinodhaka.

No akaora chinokosha zvinodhaka aiita antacid zvinodhaka, caffeine, "theophylline", "Quinidine", "propranolol", panyaya iyi, lidocaine uye "metoprolol" haina kuisa.

chaizvo kurumbidza

malignancy inofanira kunze vasati vatanga kurapwa pamwe omeprazole. Izvi imhaka yokuti kurapa ichi zvinodhaka kungavanza zviratidzo uye kunonotsa yakarurama zvokuongorora mashoko.

Pari, hapana mashoko ari matambudziko mari pamunhu anogona kudzora zvigadziriswe uye kutyaira motokari.

Mutengo uye analogues

How zvikuru ichi Anti-urikanwi zvinodhaka, se "Ortanol"? Mutengo kwezvinodhaka izvi pamusoro 100-115 rubles. For vatengi vakawanda, mari izvi zvinogamuchirika.

Chii chinogona kutsiva zvinodhaka "Ortanol"? Analogs kugadzirira ichi dzinoturwa muchimiro "omez", "Loseprazol", "Gaseka", "Omelika", "omeprazole".

Reviews

Reviews pamusoro capsules "Ortanol" akanaka kune mukuru pamwero. Varwere vanoti mushonga unoshanda antiulcer mumiririri. Rakakurumidza anobvisa chirungurira uye kunzwa kufundumwara uye nokupisa mudumbu.

Nyanzvi vanoti mushonga mu mubvunzo kunobatsirawo mararamiro zvirwere zvomudumbu turakiti chete kana kugamuchira yayo akagadzwa pedyo gastroenterologist. Vanachiremba vanotaura kuti ravo kutora mushonga uyu hakubvumidzwi, sezvo ane simba chaizvo.

Panewo yakanaka divi mishonga iyi anosanganisira ayo Kuwanikwa uye vakaderera mutengo.

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