UtanoGadziriro

"Flyuanksol": mirayiridzo kushandiswa, vanachiremba chaivo. Marwadzo "Flyuanksola" analogues zvinodhaka

Chii chinodhaka "Flyuanksol"? Mirayiridzo kushandiswa kwezvinodhaka, ayo zvinhu, marwadzo, kusunungurwa chimiro uye pharmacological zvivako zvinotsanangurwa zvizere munyaya ino. Mariri uchadzidza pamusoro zvakaitwa contraindications uye zvairatidza vakati chinodhaka, sei tinorasikirwa, chii chichaitika kana ane ovhadhozi, uye zvichingodaro. D.

The Kuronga zvinodhaka uye ayo kusunungurwa nezvimiro

Ndechipi zvinoshingaira fuma rine mishonga "Flyuanksol"? mirayiridzo kushandiswa medicament murayiridzo rinotaura kuti kutoshanda zvinoriumba izvozvo makabuda flupenthixol hydrochloride.

Kana chimiro resununguro, asi nhasi ndiye nzira dzinogona kuwanikwa bedzi madonhwe, mapiritsi uye mhinduro, mafuta anotsanangura, dzaizopiwa intramuscular yaitonga. Chokutanga mushonga iri kutengeswa muna girazi zatemennom Rine mamiririta 10, yechipiri - ari atorwa 100 kana 50 uye wechitatu - mune ampoules zvezvimedu 10.

General ehupfumi zvinodhaka

Nei mishonga "Flyuanksol"? Testimonials pamusoro mushonga uyu dzinoturwa pazasi. Mahwendefa uye jekiseni tiri boka antipsychotics. Ivo nhaka anxiolytic, antidepressant uye kunyaradza kushanda. Positive inofambiswa pamusoro zvinodhaka ichi ane ruzivo kuti zvakanyanya zvaanopa simba ari kunetsa murwere uye kunobatsira kuti mumagariro kwadzakabva.

The pharmacological zvechadenga zvinodhaka

Ndezvipi zvainyanya kuitwa pharmacological zvinodhaka "Flyuanksol"? Mirayiridzo dzokushandisa kunoratidza kuti zvinodhaka uyu neuroleptic, ichivharira adrenergic receptors uye dopamine receptors muuropi. Somugumisiro yezviri fuma kunokwanisika nyaradzo. Kazhinji, izvi zvaitika pamusoro ane 8-zuva dzose chipimo chemushonga.

Ko varwere pamusoro mishonga "Flyuanksol"? Reviews wevarwere zvine zvakawanda dzinonakidza. Kazhinji, ivo cherechedza kuti mushonga asi nokukurumidza anobvisa zviratidzo psychosis uye kuora mwoyo, uyewo zvinoita kuti kudzorerwa mafungiro. Varwere vakanga hazvina ushamwari zvinetso, muri fara nevamwe uye zvinoenderana vanhu.

Features mishonga

Sei mushonga "Flyuanksol"? Reviews vanachiremba uye dzimwe nyanzvi dzinoti zvakakurumbira zvinodhaka ichi ndechokuti, zvichienderana dose inogona kuita murwere nenzira dzakasiyana.

Antipsychotic zvazviri kunoratidza pashure medicament kushanda zvinoreva mune mari 3 MG pazuva. Nenzira, kusimba matambudziko kunowedzera chipimo chemushonga.

Huwandu 25 MG pazuva zvinodhaka hapana kunyaradza maturo. Zvisinei, zvinofanira kucherechedzwa kuti panguva dzakakwirira mishonga, zvinogona kukonzera non-chaizvo kunyaradza anokonzerwa.

Muna dose siyana yakasarudzwa neuroleptic mumiririri ane raidudzwa anxiolytic kushanda. Kana kushandisa mishonga diki (kusvika anenge 3 MG pazuva), mushonga dzingava antidepressant mishonga ine kwakajairika.

Saka, mushonga "Flyuanksol" anogona kuderedza chikuru zviratidzo psychosis, kusanganisira paranoid zvinovadadira, aone zvinhu zvisipo, uye akafunga nyonganyonga. Rine disinhibitory ehupfumi (i.e. simba uye antiautisticheskim) uye kunoderedza nedambudziko rezvinyamusi, izvo pakupedzisira inosimudzira activation varwere kuora zviratidzo, avo mumagariro kwadzakabva hwezvekukurukurirana uye kunonatsiridza sociability.

More pamusoro injectable chimiro

Kugadzirira "Flyuanksol dhepoti" ane mafuta mhinduro aiendeswa intramuscular dhepoti majekiseni. Nemamwe mashoko, mushonga uyu rakachengetedzwa fomu flupenthixol.

Kana kushandisa mhinduro iri diki uye svikiro mishonga (kusvika 100 MG ose mazuva 14) kuti murwere haasi unspecific nyaradzo. Kunyange zvazvo achiri kukura pa pamatunhu mishonga.

Chii Nyanzvi vanoti pamusoro chimiro ichi zvinodhaka ( "Flyuanksol dhepoti")? Reviews zvinopa kuti yakadai mhinduro ine refu nguva yokuwana nomurwere, pane mahwendefa mushonga. Uyezve, kutenda kwaari, zviri nyore kuti tiite chinoramba antipsychotic kurapwa, izvo zvakanyanya kukosha kuti varwere musatakura kubuda zvokurapa mushonga.

Kubva apa zvinogona vakagumisa kuti zvinodhaka "Flyuanksol dhepoti" rinogona kudzivisa kakawanda zvazvo chokuita vaingoerekana akatevedzana yokurapa. Intramuscular jekiseni anogona kuitwa panguva zvikamu zviviri kana mana mavhiki.

Pharmacokinetics

Rinhiko kunge kunyura mapiritsi "Flyuanksol"? Mushure zvokuudzwa Kutarisirwa kufadza pfungwa yezviri chinhu kunokwanisika mumaawa anenge 3-7 muna plasma. The bioavailability zvinodhaka ndiko 40%.

Active zvinodhaka chaikosha kupinda munharaunda yacho placental chipingamupinyi zvishoma. Zvinofanira kucherechedzwa kuti, riri shoma, zviri pachena chete wamai mukaka. Sezvineiwo, mashoko metabolites vane neuroleptic basa.

Sei jekiseni "Flyuanksol dhepoti"? Guide rinoti kuti pashure intramuscular jekiseni yamarudzi Kishi (Z) -flupentixol decanoate kaviri cleavage (enzymatic). Izvi anoumba zvinoshingaira chinhu pamusoro Kishi (Z) -flupentixol uye decanoic acid. The kunonyanyisa wevasungwa munguva serum iri pakutanga nokuramba pakupera vhiki yokutanga pashure jekiseni.

Kana muchigamuchira mahwendefa avo maberekero nguva iri maawa anenge 35. Kana raishandiswa mhinduro jekiseni, wevasungwa zvinoderedza exponentially ari serum (pashure 3 mavhiki).

Akaratidza kushingaira medicament ari muchimiro metabolites kuburikidza ura, neitsvo.

Zvairatidza kuti kushandiswa neuroleptic vamiririri

Mune zvimwe zviitiko, zvinodhaka rinoratidza "Flyuanksol"? chiito chacho kungava zvakasiyana, zvichienderana chipimo chemushonga.

The mushonga zvinoratidzwa pana mishonga anosvika 3 MG pazuva raitevera pathological ezvinhu:

  • mwoyo nepakati dhigirii, achiperekedzwa kuneta, kufunganya uye kushaya vanotanga;
  • psychosomatic zvirwere kuti anoratidza nemashoko asthenic siyana;
  • neurotic zvirwere (chirwere), achiperekedzwa vasingakendengi, kuora mwoyo uye kufunganya;
  • uye chenjera ezvinhu kufunganya zvinetso, uyewo mamiriro wokunzwa mupfungwa, haadi kunyaradza kana hypnotic kushanda (somuenzaniso, kana murwere ari kushandisa mapiritsi).

Medicament "Flyuanksol", analogues izvo zvichakurukurwa panopera nyaya, anogadzwa pana dosages 3 MG pazuva uye zvakawanda kana pane kutsaudzira zvinotevera: ezvinhu pfungwa dziri pamwe paranoid zvinovadadira, aone zvinhu zvisipo, nenyonganiso pamafungiro, anergy, vasingakendengi uye autism.

Contraindications pakushandisa neuroleptic vamiririri

Mune zvimwe zviitiko, haisi yakarumbidza kushandisa zvinodhaka "Flyuanksol"? Mirayiridzo yokushandisa zvinosanganisira zvinotevera mazita contraindications:

  • chevana zera (Makore 18);
  • CNS mwoyo;
  • lactation;
  • panguva pamuviri;
  • kudhaka (chenjera) barbiturates;
  • richaparara;
  • kudhaka chenjera opioid analgesics;
  • pheochromocytoma;
  • chidhakwa chenjera chepfu;
  • comatose inoti;
  • mwongo kudzvinyirira;
  • Kumwe kuchinja kunotanga muropa;
  • hypersensitivity kune neuroleptics rine tioksantenoviy marongerwo.

Zvinofanira kucherechedzwa kuti hakukurudzirwi taurira mushonga mu mishonga diki (3 MG) vachingotya wokusagadzikana kana excitations.

Drug "Flyuanksol": mirayiridzo (pamahwendefa, anosiya)

Nokuti kurapa mwoyo uye zvokuora mwoyo kwokutanga dose of medicament iri mahwendefa vanofanira kuva 1 MG kamwe pazuva (kudiwa mangwanani), kana 500 mcg kaviri daily. Kana mishonga zvazviri vasipo, uwandu zvinodhaka pavhiki kunogona ngazviwedzerwe 2 MG. Saka zuva nezuva chipimo chemushonga (2-3 MG) kukamurwa muzvikamu akawanda. Kana zvazviri vasipo kana uchishandisa mushonga ari maximal dose (i.e., 3 MG), saka zvinofanira kuregwa.

In pakurapa pfungwa ezvinhu akaisa yakawanda mishonga chete nomumwe. The kutanga daily chipimo chemushonga kunofanira 3-15 MG muna 3 yakakamurwa mishonga. Kana akakumbira, akati inzwi kunogona ngazviwedzerwe 20 kana 30 MG pazuva. The kunonyanyisa chipimo chemushonga hakufaniri anopfuura 40 MG.

Rinomiririrwa Nokuraramisa kurapwa mumiririri chinotarisirwa mune imwe mari 5-20 MG kamwe pazuva (mangwanani).

Kana donhwe "Flyuanksol", vanofanira chete kubatwa mukati. Doctors kazhinji mishonga mushonga nechimiro ichi chete nyaya kana, nokuti chero chikonzero, haagoni kutora mishonga nomuromo (piritsi). Kutsigira chipimo chemushonga varwere ndiyo 4-40 MG pazuva.

Jekiseni "Flyuanksol": kurayira, nomwoyo murefu wongororo

The jikichira mhinduro kuti intramuscular chakazara majekiseni chinofanira kupiwa zvakadzika muimba rokunze quadrant pamusoro magaro. Chipimo chemushonga uye penguva pakati kurapa vanofanira chete iiswe somunhu (hwokuzvimirira kuchirapa kushanda).

Pfungwa iyi unowanzoshandiswa nenzira imwe mari 20-40 MG (kana 1-2 Rine mamiririta) ose vhiki 2 kana 4. Zvinofanira kucherechedzwa kuti vamwe varwere kungada makuru mishonga uye pfupi penguva pakati majekiseni.

Kana akasarudzwa Vhoriyamu mushonga jekiseni (20 MG / Rine mamiririta) inopfuura 2 kana 3 Rine mamiririta kuti 1 nzira, zvakakodzera kuenda mberi pamwe chete mhinduro mukuru yevasungwa.

Preparation 100 MG / Rine mamiririta inofanira jekiseni mune bhuku 50-200 MG (kana 0.5-2 Rine mamiririta) ose 2-4 mavhiki. In chenjera kuitazve kana exacerbation chirwere dzimwe nguva zvinoda rimwe nguva sumo zvinoreva mune mari kusvika 400 MG pa zvikamu of 2 kana 1 vhiki. Mushure chenjera zviratidzo zvakaitika, unofanira kugadzira nezvishoma zvinoderedza uwandu husingakuvadzi kuti Nokuraramisa (20-200 MG ose 2-4 masvondo).

Kana kunodiwa kupfuura kubva waiita chimiro zvinodhaka nokuda parenteral kugadzirira rutsigiro kurapa, Zvinokurudzirwa kuti inobva anotevera zano:

  • daily chitsama (mu MG) zvinodhaka zviri mahwendefa X 4 = chete chipimo chemushonga (mu MG) jekiseni mazuva 14 ose.

Zvinofanira kucherechedzwa kuti mukati vhiki imwe pashure kwokubatsira mushonga vari zano kuramba kutora mushonga pamahwandefa, asi pane yakaderera dose. Tevera-up vhoriyamu uye musiyano uri pakati nzira yakatangwa maererano kuchirapa kushanda.

Kunonyanyisa chipimo chemushonga injectable mhinduro (imwe-Danho) ndiyo MG anenge 400. Saka musiyano uri pakati majekiseni kunge pane imwe vhiki.

Maererano mhinduro wevarwere, kana ikashandiswa zvakanaka, kugadzirira uye kuchengetwa zvokurapa vanorumbidza, ine kunobatsirawo hwadzo kunetsa.

nemishonga

Ko kunambwa muviri mushonga "Flyuanksol"? Marwadzo varipo vari chinodhaka, zvisinei wawo. Pano vari ikozvino.

  1. Tsinga: giperkinetiko-vane chirwere cheBP syndrome (extrapyramidal chiedza), simba, akathisia, kurukutika, dzungu, psychomotor retardation, tardive dyskinesia, dystonic siyana uye neuroleptic akaipa syndrome.
  2. Mwoyo uye ropa midziyo: tachycardia, hypotension, orthostatic.
  3. hematopoietic maitiro: granulocytopenia.
  4. Sense nhengo: kunetswa akkommodasie.
  5. GI: kupatira, jaundice cholestatic, muromo yakaoma, zvinopfuura kuchinja chiropa shanda nemiedzo.
  6. Kwemakemikari anobudiswa hurongwa: kufuta, galactorrhea, vangadikitira, gynaecomastia, kusabetsera, dysmenorrhea, wakawedzera kudya, ungaderedza libido, kupiswa.
  7. Urinary maitiro: Urinary chengetedzo.
  8. Allergies: dermatitis, photosensitivity, uye ganda nekumhanyirira.

Mirayiridzo Special kushandiswa

With Kunyatsongwarira mishonga ushandiswe varwere vane zvemwoyo zvinetso, convulsive zvirwere, kufema kukundikana, yemaziso, Parkinson, chirwere nemaronda mudumbu uye 12-tiperstnoj paura, asima, udhakwa, emphysema, Urinary chengetedzo, chiropa kukundikana, uye prostatic hyperplasia isiri yekenza.

Kana murwere kare akagamuchira neuroleptics kana tranquillizers pamwe kunyaradza chaizvoizvo, zvinokosha kurega kutora kwavari zvakanaka.

Kana mabatiro kwenguva refu, kunyanya panguva yakakwirira dosages akataura kuzvidzora uye kuyera murwere ezvinhu kuitira kugadzirisa yokuzvigadzirisa dose.

Mugore mawa pakurapwa kwechirwere cheshuga basa akati Pfungwa kungada kururamiswa yakawanda jekiseni.

In kushanda neuroleptics zvingamuka neuroleptic akaipa syndrome. chikuru Zviratidzo ayo tsandanyama Rigidity, hyperthermia, zvakachinjwa chinzvimbo mupfungwa, uye dysfunction pamusoro autonomic tsinga. Kana zviratidzo zvakadai zvinoda kukurumidza Kudzimwa kwechikwereti kugadzwa zvinodhaka uye aitsigira symptomatic kurapwa.

Kazhinji, mishonga "Flyuanksol" haakonzeri nyaradzo. Asi, pasinei ichi, zvinokosha kufunga kwadzo kukanganisa kukwanisa zvakachengeteka kushandisa muchina, kana zvimwe zvigadziriswe. Ini ndingadawo kucherechedza kuti panguva kurapa (kunyanya pakutanga), varwere vanofanira kudzivisa basa anogona nengozi (kuziva mhinduro kune mushonga).

zviitiko ovhadhozi

Kana mishonga chinobviswa zvakanaka (rakawedzerwa), zvinogona kuitika ovhadhozi. Panyaya iyi, rinoratidza zvinotevera unhu: hypo- kana hyperthermia, hope, kugwinha, extrapyramidal wenyonganyonga, kurohwa nehana, hypotension uye pakoma.

Zvokuita mumamiriro ezvinhu akadaro? Zvakakosha kuita kutsigira uye symptomatic kurapa. Kana mushonga akanga anwa, kudiwa nokukurumidza kusuka kubva mudumbu, uyewo kutora sorbent. Uyezve, zviri zvikuru kutsigira mabasa nhumbi, mwoyo uye kufema hurongwa. Hazvina varumbidzwa kushandisa epinephrine sezvo kungaita kuti BP rutapudzo. Extrapyramidal zviratidzo zvinobvira kumisa mushonga "Biperiden" uye pfari - "Diazepam".

Kudyidzana nevamwe zvinodhaka

Kana uchishandisa imwe-padanho akati medicament anogona yakakura kunyaradza anokonzerwa barbiturates, panyaya iyi, uye vamwe vamiririri vane inhibitory zvainoita CNS.

Kugadzirira "Flyuanksol" haisi varumbidzwa kushandisa pachiimbwa guanethidine uye Drug chete ndozvinoitawo. Izvi imhaka yokuti antipsychotics anogona chaizvo simba ravo antihypertensive migumisiro.

With chete-kushandiswa medicament "Flyuanksol" inogona kuderedza efficacy zvinodhaka "levodopa" uye dzimwe adrenergic nevamiririri.

Panguva iyoyowo achitora zvinodhaka ane "piperazine" uye "MCP" Sezvineiwo kunowedzera ngozi yokubatwa extrapyramidal rebipolar.

Zvinofanira kucherechedzwa kuti neuroleptic chinodhaka anounzwa kugadzirisa kuti jekiseni chero zvazvingava harifaniri kuvhenganiswa nemamwe zvinwiwa.

Price uye analogues zvinodhaka

How kuzhinji chinodhaka "Flyuanksol"? mutengo wayo zvakakwirira zvikuru. Saka, nokuti mahwendefa 1 MG penyu 50 vanofanira kubhadhara anenge 500 rubles Russian. Kana uchida 100 5 MG pamahwendefa, vanogona kutenga kuti 1,200 rubles. Kana injectable chimiro chinodhaka, chinotova anodhura. Over 10 ndiro (20 MG / Rine mamiririta) vemishonga zvinoda anenge 2300 rubles.

Zvakadini kana murwere haakwanisi kutenga mushonga "Flyuanksol"? analogues Its vanotengeswa mune zvinenge zvose chemishonga ngetani. Pakati pavo pane zvinotevera:

  1. Kugadzirisa "Flyuanksol dhepoti". Zviri nokukurumidza uye kupfuura simba zvinodhaka. Zvisinei, zviri pamahwendefa zvikuru zvinodhura.
  2. "Klopiksol" mishonga. In ukoshi riri pedyo chaizvo chepakutanga. It anoenderera mberi Sale pamahwendefa uye ane contraindications shoma.
  3. "Truksal" zvinoreva. Inotengeswa pamahwendefa. Huru nani vachifarira kushandiswa kwayo vana vane 3-makore. Arasikirwe zvishoma pamusoro chepakutanga.

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