Utano, Kugadzirira
Kugadzirira "Algezir Ultra": mirayiridzo yekushandiswa, tsanangudzo, kuumbwa nekuongororwa
Munguva ichangopfuura, vanachiremba vanowanzogadza varwere "Algesir Ultra". Iyo mirayiridzo yeiyo chigadziro inonyatsodzidzisa uye inotsanangura zvinoshandiswa pakushandisa kwayo kumapoka akasiyana-siyana evarwere, asi haigadziri ruzivo rukuru pamusoro pekuti iyo sarudzo inoshanda sei mumuviri.
Pharmacology
Mukugadzirwa kwechirwere-NSAID, iyo inotora naphthylpropionic acid. Mukuita kwekutora ichi chirwere chinopesana nekuputika, antipyretic, pamwe nekufananidzira, izvo zvinowanzoratidzwa nekuongorora pamusoro pe "Algesir Ultra." Iyo mirayiridzo yechishandiso inoratidzawo mavara aya.
Iyo nzira yekuita kwechirwere ichi inowirirana zvakananga nekudzivirirwa kwe enzyme chaiyo COX, iyo inoita kuti zvikwanise kudzvinyirira kushandiswa kwe prostaglandids kubva kune arachidonic acid sezvinogona kubudirira. Uyezve, uyu mujeri anopa kubviswa kwe platelet aggregation.
Kunyatsotarirwa kunofanira kubhadharwa kune chokwadi chokuti panguva yekushandiswa kwemishonga inorwadza chirwere chinoderera, kusanganisira kurwadziwa kwepamuviri pamwe chete nekufamba uye kuzorora. Muchigadziriro chokubvuma kuputika kwemajoini kunoderera, kuoma kwemangwanani, kuwedzera kwekufamba kunowedzera, iyo inowanikwa nevose vanenge vakasiya mhinduro pamusoro peAlgesir Ultra. Iyo mirayiridzo inewo ruzivo rwakadaro, asi inotaurawo kuti kupesana-kupisa simba kunogona kuitika pakuguma kwevhiki yekutanga yekushanda.
Pharmacokinetics
Zvadaro, kutora iyi mishonga mukati napapapisi inotanga kukurumidza kukurumidza kubva pamigwagwa yekudya. IC max mu plasma inotanga kuongororwa kare kwemaawa mana mushure mekutonga. Izvo zvinofanira kuonekwa kuti kushandiswa panguva imwechete kwechirwere ichi nechikafu kunogona kuderedza kutengesa kwekudya, asi hakunoderedzeri kubatwa kwehuwandu. Nhamba yepamusoro inopesana nekunakidza kwakanaka munyaya yehutongi hwehutongi, asi munyaya ino kune kunonoka kunonoka, kana ichienzaniswa nekuisa.
Mukurapa kwekurapa, ichi chinosunga kumapuroteni e plasma anenge anenge 100%. Kuwedzera kwepasmaxen mumapulama kunowedzera zvakaenzana mukushandiswa kwemasero kusvika 500 mg, asi pavanowedzera kuwedzerwa kune kuwedzerwa kwebvumirano, iyo inokonzerwa nekuzadzwa kwakakwana kweprotini ye plasma.
Naproxen inopinda mukati me synovial fluid.
T 1/2 inenge maawa gumi nemaviri. Inenge 95% yehuwandu hwemuti uyu inogadziriswa mumamiriro ekushandura emuti, 6-O-desmethylnaproxen uye maitiro ayo akasiyana-siyana. Zvose zvese munguva yemberi iri mberi mushure mekugamuchira kwacho zvakasvibiswa nemasese.
Dosage
Zvakakosha kuziva kuti zvinokurudzirwa kuti munhu mumwe nomumwe aenzaniswe nehutano hwehutano hwechirwere mumurwere. Kugadzirira "Algesir Ultra" murayiridzo unoti vanhu vakuru vanorayirwa kuitora pamadhora e 0.5-1 g pazuva pazuva rekuparadzanisa, asi chiitiko chezuva nezuva chekugadzirisa chirwere chemazuva ose chinofanira kunge chiri mamiriyoni 500.
Zvose zvinogona kuitika zuva rega rega 1.75 g.
Nhamba yevana
Kana kurapwa kuchiitwa kune varwere vane makore 1 kusvika ku5, zvino munyaya iyi vanofanira kushandisa 2.5-5 mg pamakilogiramu pazuva kwema 1-3 madhora zuva rega rega, nepamusoro pekugona kurapwa munyaya iyi inogona kuva 14 Mazuva. Mukurapa kwevana vechirwere muvana vaduku vanopfuura makore mashanu, chirwere chezuva nezuva chakasimbiswa uye chinonzi 10 mg nekg.
Kupindira kwemishonga kwe "Algezir Ultra"
Mirayiridzo yekushandiswa inoti kana iyo inoshandiswa panguva imwe chete neine antacids, iyo inosanganisira aluminium uye magnesium, pamwe ne-sodium bicarbonate, zvino munyaya iyi inoshungurudza zvakanyanya kudyiwa kwe naproxen, iyo inonyanya kukosha mukurapa.
Kana iyo sarudzo inoshandiswa pamwe chete neanticoagulants isinganzwisisiki, ipapo pane zvingangodaro zvigadziriswe pamigumisiro yemishonga iyi, iyo yakaonekwa mukugadzira zvidzidzo zvekliniki dzakananga.
Uyewo mukugadzirisa kwekuita zvidzidzo, zvakagadziriswa kushandiswa panguva imwe chete kwechirwere ne amoxicillin zvakadzidzwa, izvo zvakaguma mukugadzirwa kweNephrotic syndrome mune dzimwe mamiriro ezvinhu . Kana "Algesir Ultra" yakashandiswa neacetylsalicylic acid, mune dzimwe nguva misi yose ye naproxen mu plasma yeropa yakaderera.
Zvimwe zvikamu zvekubatana
Pakati pezvimwe zvinhu, zvakakosha kucherechedza mimwe mimwe mamiriro ezvinhu, izvo zvinoratidzwa mumirairo yekugadzirira "Algesir Ultra" (mahwendefa):
- Nechishandiswa panguva imwe chete, kukwanisa kweimwe shanduko mu pharmacokinetic miganhu ye diazepam inopiwa;
- Kana iyo sendimi yakashandiswa panguva imwechete ne caffeine, mhizha ye naproxen inogona kuwedzerwa;
- Kana ichibatanidzwa ne lithium carbonate , zvinokwanisika kuwedzera kuwanda kwe lithiamu muropa plasma;
- Kusanganiswa ne methotrexate kunowedzera kuwedzerwa kwehutu hweiyo chinhu;
- Apo "Algezir Ultra" inoshandiswa panguva imwechete ne probenecid, musanganiswa wose we naproxen mu plasma yeropa yakaderedzwa;
- Kushanda pamwe chete nesaricylamide kunoita kuti zvikwanise kuwedzera chiito cheiyo chinhu.
Iko kune ruzivo runoratidza kuti kana chirwere ichi chinoshandiswa zvakagadzikana ne morphine, pakupedzisira icho chinogona kutungamirira kukurudzirwa kwemyoclonus. Uyewo, pamwe chete nekushandiswa pamwe chete ne prednisolone, kune kuwedzera kukuru muhuwandu hwekufungidzirwa kweiyi muropa re plasma. Mukuwedzera, panewo kushandiswa panguva imwe chete ne furosemide, iyo inopa kuderera kwechiito chekuita kwechirwere chechigadzirwa ichi. Iyo inoratidzwa nezvechigadzirwa chakadai segadziriro "Algesir Ultra", kuongororwa. Iyo mirayiridzo inoratidzawo chiitiko ichi chemishonga.
Kubata uye kubata
Zvinokurudzirwa kushandisa mishonga iyi nekuchenjerera kwakanyanya mumadzimai ane pamuviri kana kuti anokanganisa, uye kunyanya izvi zvinoshanda kune avo varipo panguva yekutanga kana yechitatu mitatu. Chinhu apa ndechokuti mushure mokutora ichi chinopisa mishonga chinodhaka chinotanga kupinda mukati mechigadziro chinoputika, uye chinozobudiswa zvishoma zvishoma nemukaka wemvere.
Zvikanganiso
Inofanira kuve yakarongerwa mitemo yakawanda, iyo inoratidza kugadzirira "Algesir Ultra" mirayiridzo yekushandisa. Tsanangudzo munyaya ino inopiwa mazvikwata akasiyana-siyana emitumbi:
- Kugadzirisa chirwere. Mukati yekugamuchirwa, panogona kuva nekurutsa, kusuruvara, kunzwa kusagadzikana munharaunda yepigastric. Muzviitiko zvisingawanzoitiki, pane zvipembenene zvinokonzera uye zvironda zvegumbo rekudya, pamwe nekuputsika kwakasiyana kwechiropa chinoshanda nekubuda ropa.
- Central nervous system. Paunenge uchishandisa mushonga mune vamwe varwere, kurara, kuora musoro, pamwe nekuderedza kushanya kwepfungwa dzepfungwa. Muzviitiko zvisingawanzoitiki, kushandisa chigadzirwa ichi, kune kusiyana kwakasiyana-siyana kwekunzwa, sezvinoratidzwa nemirayiridzo "Algesir Ultra" mirayiridzo yekushandiswa. Izvo zvinyorwa hazvitsananguri zvakajeka ichi chinhu chekushandiswa.
- The hematopoiesis system. Kunyanya kushandiswa kwechirwere ichi kunotungamirira kune zvinoitika zve granulocytopenia uye thrombocytopenia, uye hemolytic kana aplastic anemia.
- Kuporesa. Muzviitiko zvisingawanzoitiki, pineumonia isina simba inogona kukura .
- Urinary system. Muzviitiko zvisingawanzoitiki, zvakasiyana-siyana zvinokonzerwa nehupombwe zvinogona kuitika.
- Allergic reaction. Mune rimwe boka revarwere, urticaria, kuputika kweganda uye edema yaQuincke yakaonekwa panguva yekudzidza, iyo inowanzoita zvirwere zvinokonzerwa neanoric reaction kune zvakasiyana-siyana zvinoumba mishonga, sezvinotaurwa mu "Algesir Ultra" mirayiridzo yekushandisa. Mishonga munyaya ino haigone kumira.
Pakati pezvimwe zvinhu, zvinokodzera kunyatsotarisirwa kuti mune zvakaitika pamagetsi, kune ngozi yekuvhara mucoid nehutachiona husina kuchena kana kuonekwa kwekuzvidzivirira kunorwadza.
Inoshandiswa rini?
Mumakore mashomanana apfuura, vanachiremba vemazuva ano vawanzotanga kuronga iyi mishonga kuvarwere vavo panguva yekurapwa kwezvirwere zvakasiyana-siyana, kusanganisira izvo zvinotsanangura mazano ekushandiswa kweAlgesir Ultra. Mutengo wezvinodhaka uyu unokwanisika kusvika kumunhu wose, uye naizvozvo inorayirwa kakawanda panzvimbo yehuwandu hwemamwe maitiro akafanana.
Kunyanya, zvakakodzera kucherechedza zvirwere zvakawanda zvakakura, mukurapa iyo inoshandiswa kunyanya kushingaira:
- Osteoarthritis;
- Rheumatoid arthritis;
- Ankylosing spondylitis;
- Kuwedzera kwegout;
- Articular syndrome;
- Neuralgia;
- Myalgia;
- Pain in the spine;
- Kushungurudzika kuputika kwezvinyama zviduku kana musishusekeletal system.
Pakati pezvimwe zvinhu, "Algesir Ultra" inowanzowanikwa semubatsiri pakurapa zvirwere zvakasiyana-siyana zvinotapukira uye zvinoputika zvezvikamu zve ENT, primary dysmenorrhea, adnexitis, pamwe nemazino nemusoro.
Contraindications
Kune zviitiko zvakasiyana-siyana umo chigadzirwa ichi hachibvumirwi kushandiswa, uye izvi zvinoratidza "Algesir Ultra" yekugadzirira mazano pamusoro pekushanda (tsanangudzo). Vanachiremba vanoongorora zvakare vanowanzoratidza kuti ichi chirwere hachina kukurudzirwa kuti chishandiswe mumamiriro ezvinhu anotevera:
- "Aspirin triad";
- Mhando dzose dzezvipembenene zvinokonzera uye zvekuonda mumutsara wepamuviri;
- Akarondedzera kushungurudzwa mumabasa eitsvo;
- Kupesana kwehematopoiesis system;
- Anodudzira kusagadzikana mumabasa echiropa;
- Kunyanya kunzwisisika kune naproxen nezvimwe zvinhu izvo chikamu chechirwere ichi.
Pakati pezvimwe zvinhu, kushandiswa kwemugadziro uyu hakurudzirwi kune vana pasi pezera remakore, sekuratidzwa nemirayiridzo ye "Algesir Ultra" mirayiridzo. Mutengo wechigadzirwa ichi 85-90 rubles. Kwepiritsi gumi.
Special instructions
Kunyanya kuchenjerera iyi iyi inofanira kushandiswa mukurapwa kwezvirwere zvakasiyana-siyana zveitsvo uye chiropa, chirwere chepamuviri munhoroondo, pamwe nekushaya mwoyo, hypertension kana kuvapo kwezvirwere zvinotapira. Kunyanya, inofanirwa kuve yakagadzirirwa kutarisana nachiremba kuti kana mushonga wacho unogona kushandiswa pakugadzirisa kukuru kwekuvhiya.
Muchirapa inofanira kugara ichichengetedza kugadzirisa kushanda kwetsvo uye chiropa, pamwe chete nemufananidzo wehutachiona ropa. Kana zvakakosha kuziva kuti chiyero chema-17-ketosteroids, kudya kwe naproxen kunofanira kuregererwa maawa makumi maviri isati yasati yasvika.
Kunyatsoteerera kunofanira kubhadharwa kuitika kuti kutora mushonga uyu kunobata kukwanisa kutyaira motokari uye kugadzirisa nzira dzakasiyana-siyana. Munyaya iyi, zvakanakisisa kuti urege kubva kune zvingangoita zvinhu zvine ngozi zvakananga zvakananga nekudiwa kwekutarisa kwekucherechedza uye kukurumidza kukurumidza kwekuita kwepfungwa, apo "Algezir Ultra" iri kushandiswa. Mirairo yekushandiswa pamushonga wega wega inotsanangura pfungwa iyi.
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